PHD-IN-1
PHD-IN-1 (compound 80) is a potent inhibitor of PHD2,with an IC50 value of ≤5 nM. PHD-IN-1 shows EC50s of 2.5 μM in EPO Elisa assay both in Caco2-HIFla-HiBiT-clone-1 cells and Hep3B cells,respectively.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 2924182-31-8
- Fòrmula: C24H23N7O2
- Peso molecular:441.49
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
IC50: ≤5 nM (PHD2)[1]
Chemical Information
-
No. CAS 2924182-31-8
-
Peso molecular 441.49
-
Fòrmula C24H23N7O2
-
SMILES
OC1=C(C(NCC2=CN=C(C#N)C=C2)=O)N=CC3=C1C=CC(N4[C@]5([H])CN(C6CC6)[C@](C5)([H])C4)=N3
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)