1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. HIF/HIF Prolyl-Hydroxylase
  4. HIF/HIF Prolyl-Hydroxylase Inhibitors

HIF/HIF Prolyl-Hydroxylase Inhibitors

HIF-1α

HIF

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

HIF/HIF Prolyl-Hydroxylase Inhibitors, Agonists, Activators & Degraders
상품명 HIF-1α HIF Purity
Beta-Sitosterol (purity>98%)
HIF-1α
  99.74%
Cryptochlorogenic acid
HIF-1α
  99.87%
Bavachinin  
HIF-1α
99.95%
Deoxyshikonin  
HIF-1α
HIF-1β
99.96%
TP0463518  
HIF-2α
99.25%
VHL-IN-1
HIF-1α
  99.84%
iGP-1
HIF-1α
  99.43%
Streptonigrin
HIF-1α
  99.20%
GW-405833
HIF-1α
  98.91%
Dendrophenol
HIF-1α
  99.93%
Pseudolaric Acid B
HIF-1α
  99.47%
Cephalomannine
HIF-1α
  99.04%
GW405833 hydrochloride
HIF-1α
  99.59%
PROTAC HIF-1α degrader-1
HIF-1α, IC50: 7.54 μM
  98.02%
Izilendustat
HIF-1α
HIF-2
98.01%
Iminostilbene
HIF-1α
  99.34%
Bendazol
HIF-1α
  99.60%
AG01
HIF-1α
 
NEO-811  
HIF-1β
RH01504  
HIF-2α, Kd: 5.42 nM
T7117
HIF-1α
 
Cyclo(CRLLIF)  
HIF-2α, Kd: 10.2 μM
HIF-1α, Kd: 14.5 μM
L-Glutamine (GMP)
HIF-1α
 
HIF-2α-IN-17  
HIF-2α
HIF-2α-IN-18  
HIF-2α, IC50: 8.1 nM
Cryptolepine
HIF-1α
 
HIF-1α-IN-8
HIF-1α, IC50: 2.02 μM
 
KST012174 hydrochloride
HIF-1α
 
Anti-inflammatory agent 79
HIF-1α, IC50: .55 μM ([1])
 
ZG-2686  
HIF-2α, EC50: 0.25 μM
PROTAC HIF-1α degrader-2
HIF-1α, DC50: 22.4 μM
 
HIF-1α-IN-10
HIF-1α
 
CHNQD-03301
HIF-1α, IC50: 10.97 nM
 
PHD2-IN-4
HIF-1α
 
D-01
HIF-1α, IC50: 4.86 μM
 
Cyclo(CRVIIF)  
HIF-1α, Kd: 65 μM
HIF-2α, Kd: 123 μM
HATC
HIF-1α
 
O-Carboranylphenoxyacetanilide
HIF-1α