1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. HIF/HIF Prolyl-Hydroxylase
  4. HIF/HIF Prolyl-Hydroxylase Inhibitors

HIF/HIF Prolyl-Hydroxylase Inhibitors

HIF-1α

HIF

PHD1

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

HIF/HIF Prolyl-Hydroxylase Inhibitors, Agonists, Activators & Degraders
Product Name HIF-1α HIF PHD1 Purity
PX-478
HIF-1α
    99.58%
Beta-Sitosterol (purity>98%)
HIF-1α
    99.74%
Cryptochlorogenic acid
HIF-1α
    99.87%
Deoxyshikonin  
HIF-1α
HIF-1β
  99.96%
Bavachinin  
HIF-1α
  99.95%
TP0463518  
HIF-2α
  99.25%
IDF-11774
HIF-1α
    99.30%
iGP-1
HIF-1α
    99.43%
VHL-IN-1
HIF-1α
    99.84%
Streptonigrin
HIF-1α
    99.20%
GW-405833
HIF-1α
    98.91%
Dendrophenol
HIF-1α
    99.93%
Pseudolaric Acid B
HIF-1α
    99.47%
Cephalomannine
HIF-1α
    99.04%
GW405833 hydrochloride
HIF-1α
    99.59%
PROTAC HIF-1α degrader-1
HIF-1α, IC50: 7.54 μM
    98.02%
Iminostilbene
HIF-1α
    99.34%
Izilendustat
HIF-1α
HIF-2
  98.01%
Bendazol
HIF-1α
    99.60%
AG01
HIF-1α
   
NEO-811  
HIF-1β
 
RH01504  
HIF-2α, Kd: 5.42 nM
 
Caulerpin
HIF-1α
   
T7117
HIF-1α
   
Cyclo(CRLLIF)  
HIF-2α, Kd: 10.2 μM
HIF-1α, Kd: 14.5 μM
 
SH-26    
PHD1
L-Glutamine (GMP)
HIF-1α
   
HIF-2α-IN-17  
HIF-2α
 
HIF-2α-IN-18  
HIF-2α, IC50: 8.1 nM
 
Cryptolepine
HIF-1α
   
HIF-1α-IN-8
HIF-1α, IC50: 2.02 μM
   
KST012174 hydrochloride
HIF-1α
   
Anti-inflammatory agent 79
HIF-1α, IC50: .55 μM ([1])
   
ZG-2686  
HIF-2α, EC50: 0.25 μM
 
PROTAC HIF-1α degrader-2
HIF-1α, DC50: 22.4 μM
   
HIF-1α-IN-10
HIF-1α
   
CHNQD-03301
HIF-1α, IC50: 10.97 nM
   
PHD2-IN-4
HIF-1α
   
D-01
HIF-1α, IC50: 4.86 μM
   
Cyclo(CRVIIF)  
HIF-1α, Kd: 65 μM
HIF-2α, Kd: 123 μM
 
HATC
HIF-1α
   
PX-478 free base
HIF-1α
   
PX-478 (Standard)
HIF-1α
   
MPT0B098
HIF-1α
   
O-Carboranylphenoxyacetanilide
HIF-1α