1. GPCR/G Protein
  2. Protease-Activated Receptor (PAR)
  3. Parmodulin 2

Parmodulin 2 (Synonyms: ML161)

Cat. No.: HY-13965
Handling Instructions

Parmodulin 2 (ML161),a probe, is an allosteric inhibitor of protease-activated receptor 1 (PAR1) with an IC50 of 0.26 μM. Parmodulin 2 inhibits platelet aggregation induced by a PAR1 peptide agonist or by thrombin and has shown cytoprotective effects[1, 2].

For research use only. We do not sell to patients.

Parmodulin 2 Chemical Structure

Parmodulin 2 Chemical Structure

CAS No. : 423735-93-7

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Description

Parmodulin 2 (ML161),a probe, is an allosteric inhibitor of protease-activated receptor 1 (PAR1) with an IC50 of 0.26 μM. Parmodulin 2 inhibits platelet aggregation induced by a PAR1 peptide agonist or by thrombin and has shown cytoprotective effects[1, 2].

IC50 & Target

PAR1[1]

Molecular Weight

361.23

Formula

C₁₇H₁₇BrN₂O₂

CAS No.

423735-93-7

SMILES

O=C(NC1=CC=CC(NC(CCC)=O)=C1)C2=CC=CC=C2Br

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Parmodulin 2
Cat. No.:
HY-13965
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