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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
11 Results for "
B1R
" in MedChemExpress (MCE) Product Catalog:
Products (11)
11 Results for "B1R" in MCE Product Catalog:
Cat. No.: HY-100013B1R
CAS No.: 1609563-70-3
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(1S,2S)-2-PCCA (hydrochloride) (Standard) is the analytical standard of (1S,2S)-2-PCCA (hydrochloride) (HY-100013B1). This product is intended for research and analytical applications. (1S,2S)-2-PCCA hydrochloride is a less active diastereomer of 2-PCCA. 2-PCCA is a GPR88 receptor agonist, and inhibits GPR88-mediated cAMP production, with an EC50 of 116 nM in HEK293 cells.
Cat. No.: HY-W704574
CAS No.: 77102-28-4
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Mergetpa is a reversible Arg-carboxypeptidase inhibitor with high affinity. Mergetpa reduces B1R. Mergetpa blocks the overexpression of IL-1β protein and mRNA in glucose-fed rats. Mergetpa significantly increases the expression of IL-1β protein in the renal cortex. Mergetpa is used to block the conversion of kinins and B2 receptor antagonists into metabolites lacking the C-terminal arginine. Mergetpa inhibits the time-dependent enhancement of the response of isolated rabbit aorta to bradykinin. Mergetpa preserves the chemotactic activity of full-length SDF-1α on cells. Mergetpa reverses hyperglycemia, excessive weight gain, elevated levels of oxidative stress markers and overexpression of inflammatory markers in glucose-fed rats [1] .
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Cat. No.: HY-P3209
CAS No.: 115035-45-5
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Cat. No.: HY-P5518A
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Cat. No.: HY-P5518
CAS No.: 1054763-33-5
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Cat. No.: HY-RS01454
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BDKRB1 Human Pre-designed siRNA Set A contains three designed siRNAs for BDKRB1 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS01455
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Bdkrb1 Mouse Pre-designed siRNA Set A contains three designed siRNAs for Bdkrb1 gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-P706112
Purity: ≥ 85%, as determined by reducing SDS-PAGE.
Synonyms: VRK2; VRK Serine/Threonine Kinase 2; Serine/Threonine‑Protein Kinase VRK2; Vaccinia Related Kinase 2; Vaccinia‑Related Kinase 2; Vaccinia Virus B1R‑Related Kinase 2
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Cat. No.: HY-P77504
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: VRK1; VRK Serine/Threonine Kinase 1; Serine/Threonine‑Protein Kinase VRK1; Vaccinia Related Kinase 1; Vaccinia‑Related Kinase 1; Non‑Specific Serine/Threonine Protein Kinase; Vaccinia Virus B1R‑Related Kinase 1; HMNR10; PCH1A; PCH1
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Cat. No.: HY-P706111
Purity: ≥ 85%, as determined by reducing SDS-PAGE.
Synonyms: VRK1; VRK Serine/Threonine Kinase 1; Serine/Threonine‑Protein Kinase VRK1; Vaccinia Related Kinase 1; Vaccinia‑Related Kinase 1; Non‑Specific Serine/Threonine Protein Kinase; Vaccinia Virus B1R‑Related Kinase 1; HMNR10; PCH1A; PCH1
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
