8 Results for "

Endomorphin

" in MedChemExpress (MCE) Product Catalog:
Products (8)

8 Results for "Endomorphin" in MCE Product Catalog:

3
Endomorphin 1
Endomorphin 1
0 Images
3 Cited Publications
Cat. No.: HY-P0185
CAS No.: 189388-22-5
Category:  

Natural Products Monophenols Pyrrole Alkaloids Neurological Disease Phenols Endogenous metabolite Disease Research Fields Indole Alkaloids

Target:  

Opioid Receptor

Endomorphin 1, a high affinity, highly selective agonist of the μ-opioid receptor (Ki: 1.11 nM), displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Endomorphin 1 has antinociceptive properties .
3
Endomorphin 1 acetate
Endomorphin 1 acetate
0 Images
3 Cited Publications
Cat. No.: HY-P0185A
CAS No.: 1276123-71-7
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Endomorphin 1 acetate, a high affinity, highly selective agonist of the μ-opioid receptor (Ki: 1.11 nM), displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Endomorphin 1 acetate has antinociceptive properties .
Acetyl tetrapeptide-15
Acetyl tetrapeptide-15
0 Images
Cat. No.: HY-P1626
CAS No.: 928007-64-1
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Acetyl tetrapeptide-15 is a synthetic peptide. Acetyl tetrapeptide-15 is derived from endomorphin-2 (Tyr-Pro-Phe-Phe-NH2), a human μ-opioid agonist with selective anti-nociceptive effect. Acetyl tetrapeptide-15 reduces skin hyperreactivity producing inflammatory, chronic and neuropathic pain, by increasing the threshold of neuronal excitability in μ-opioid receptor via an endorphin-like pathway. Acetyl tetrapeptide-15 is used in the cosmetics for sensitive skin .
BMS-986187
BMS-986187
0 Images
Cat. No.: HY-120613
CAS No.: 684238-37-7
Purity:  99.66%
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

BMS-986187 is an δ-opioid receptor-selective positive allosteric modulator (PAM) with an EC50 of 0.03 μM and a pKB of 6.02 (～1 μM). BMS-986187 has no observable PAM activity at the μ-receptor (EC50=3 μM) .
Endomorphin 2 TFA
Endomorphin 2 TFA
0 Images
Cat. No.: HY-P0186A
CAS No.: 1276124-00-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM .
Endomorphin 2
Endomorphin 2
0 Images
Cat. No.: HY-P0186
CAS No.: 141801-26-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Endomorphin 2, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.
N-terminally acetylated Endomorphin-1
N-terminally acetylated Endomorphin-1
0 Images
Cat. No.: HY-P1171
CAS No.: 936000-56-5
Synonyms: Ac-L-Tyr-L-Pro-L-Trp-L-Phe-CONH2
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.
2-Aminodecanoic acid
2-Aminodecanoic acid
0 Images
Cat. No.: HY-W099633
CAS No.: 17702-88-4
Target:  

Amino Acid Derivatives

Research Areas:  

Neurological Disease

2-Aminodecanoic acid is a lipophilic α-amino acid with an aliphatic side chain of 10 carbon atoms. 2-Aminodecanoic acid modifies the N-terminus of endogenous opioid peptide endomorphin-1 to enhance metabolic stability and membrane permeability. 2-Aminodecanoic acid can be used for the research of neuropathic pain .
Assay Types