1. GPCR/G Protein
    Neuronal Signaling
  2. Opioid Receptor
  3. Endomorphin 2 TFA

Endomorphin 2 TFA 

Cat. No.: HY-P0186A Purity: 98.72%
Handling Instructions

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.

For research use only. We do not sell to patients.

Endomorphin 2 TFA Chemical Structure

Endomorphin 2 TFA Chemical Structure

CAS No. : 1276124-00-5

Size Price Stock Quantity
10 mM * 1 mL in Water USD 127 In-stock
Estimated Time of Arrival: December 31
5 mg USD 84 In-stock
Estimated Time of Arrival: December 31
10 mg USD 144 In-stock
Estimated Time of Arrival: December 31
25 mg USD 312 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of Endomorphin 2 TFA:

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Description

Endomorphin 2 TFA, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM[1].

IC50 & Target

Ki: 20-30 nM (kappa3 opioid receptor)[1]

Molecular Weight

685.69

Formula

C₃₄H₃₈F₃N₅O₇

CAS No.

1276124-00-5

SMILES

O=C(N)[[email protected]](CC1=CC=CC=C1)NC([[email protected]](CC2=CC=CC=C2)NC([[email protected]]3N(C([[email protected]](CC4=CC=C(C=C4)O)N)=O)CCC3)=O)=O.OC(C(F)(F)F)=O

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -80°C 2 years
  -20°C 1 year
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

H2O : 62.5 mg/mL (91.15 mM; Need ultrasonic)

DMSO : < 1 mg/mL (insoluble or slightly soluble)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.4584 mL 7.2919 mL 14.5838 mL
5 mM 0.2917 mL 1.4584 mL 2.9168 mL
10 mM 0.1458 mL 0.7292 mL 1.4584 mL
*Please refer to the solubility information to select the appropriate solvent.
References
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Endomorphin 2 TFA
Cat. No.:
HY-P0186A
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