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Substrate Analogue Inhibitors

" in MedChemExpress (MCE) Product Catalog:
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Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-19593
    Nikkomycin Z
    2 Publications Verification

    		 Fungal Infection
    Nikkomycin Z is a nucleoside peptide and an orally active antifungal agent. Nikkomycin Z inhibits chitin synthesis by acting as a competitive analogue of the chitin synthase substrate UDP-N-acetylglucosamine. Nikkomycin Z has antifungal activity .
    Nikkomycin Z
  • HY-W104477
    3-Fluoro-L-tyrosine

    		Others Metabolic Disease
    3-Fluoro-L-tyrosine is a tyrosine analogue, inhibits transamination by tyrosine aminotransferase (TAT). And 3-FluoroL-tyrosine has been shown to be biologically incorporated into proteins in place of tyrosine. 3-Fluoro-L-tyrosine pretends to be the substrate of rat liver tyrosine aminotransferase, markedly disturbs the Tyr-TAT association .
    3-Fluoro-L-tyrosine
  • HY-19548
    BEC

    		Arginase Endocrinology
    BEC, an arginine analogue, is a slow-binding competitive inhibitor of the binuclear manganese metalloenzyme arginase. BEC enhances substrate flux to NO synthase, thereby enhancing NO-dependent smooth muscle relaxation in the corpus cavernosum, and enhances penile erection .
    BEC
  • HY-W396889
    (R)-N-(1-Hydroxypropan-2-yl)palmitamide

    		Phospholipase Inflammation/Immunology
    (R)-N-(1-Hydroxypropan-2-yl)palmitamide (compound 24) is a substrate analog inhibitor of phospholipase A2 .
    (R)-N-(1-Hydroxypropan-2-yl)palmitamide
  • HY-131812
    5'-dAMPS

    2'-Deoxyadenosine 5'-O-thiophosphate

    		 Nucleoside Antimetabolite/Analog Others
    5'-dAMPS is an analogue of 5'-dAMP and thus a potential substrate, competitive inhibitor or regulator of enzymes that interact with dAMP .
    5'-dAMPS
  • HY-131810
    5'-AMPS

    		Nucleoside Antimetabolite/Analog Others
    5'-AMPS is an analogue of 5'-AMP and a substrate and competitive inhibitor or regulator of enzymes that interact with 5'-AMP .
    5'-AMPS
  • HY-131813
    5'-dCMPS

    2'-Deoxycytidine-5'-O-monophosphorothioate

    		 Drug Derivative Others
    5'-dCMPS is an analogue of 5'-dCMP and a potential substrate, competitive inhibitor or regulator of enzymes that interact with 5'-dCMP .
    5'-dCMPS
  • HY-131815
    5'-dIMPS

    		Nucleoside Antimetabolite/Analog Others
    5'-dIMPS is an analogue of 5'-dIMP and a potential substrate, competitive inhibitor or regulator of enzymes that interact with 5'-dIMP .
    5'-dIMPS
  • HY-131814
    5'-dGMPS

    		Nucleoside Antimetabolite/Analog Others
    5'-dGMPS is an analogue of 5'-dGMP and a potential substrate, competitive inhibitor or regulator of enzymes that interact with 5'-dGMP .
    5'-dGMPS
  • HY-131817
    5'-GMPS

    		DNA/RNA Synthesis Others
    5'-GMPS is an analogue of 5'-GMP and a substrate, competitive inhibitor or regulator of enzymes that interact with 5'-GMP. 5'-GMPS is suitable as a primer of RNA synthesis by T7 RNA polymerase .
    5'-GMPS
  • HY-156455
    SETD7-IN-1

    		Histone Methyltransferase Cancer
    SETD7-IN-1 (compound 7) is a PFI-2 (HY-18627) analogue. SETD7-IN-1 is a substrate and inhibitor of histone lysine methyltransferase SETD7, with an IC50 of 0.96 ± 0.10 µM .
    SETD7-IN-1
  • HY-137744
    MANT-GppNHp

    		Adenylate Cyclase Nucleoside Antimetabolite/Analog Infection
    MANT-GppNHp is a competitive adenyl cyclase (AC) inhibitor. MANT-GppNHp is a fluorescently labeled GTP (HY-113225) analogue. MANT-GppNHp interacts with the hydrophobic pocket near the AC catalytic site through its MANT group, thereby directly blocking the binding of the substrate ATP. MANT-GppNHp can be used to study diseases related to the increased activity of AC (such as cholera) .
    MANT-GppNHp
  • HY-W879508
    ALT-2074

    BXT-51072

    		 Cytochrome P450 Glutathione Peroxidase Inflammation/Immunology
    ALT-2074 (BXT-51071) is an orally active catalytic analogue of glutathione peroxidase. ALT-2074 is an inhibitor of human CYP3A, with its IC50 value ranging from 2.0 to 2.6 μM. ALT-2074 shows only a weak inhibitory effect on CYP3A in vivo, suggesting that it may not significantly affect the metabolism of CYP3A substrate drugs. ALT-2074 can be used to study inflammatory diseases characterized by reactive oxygen species, such as acute coronary syndrome .
    ALT-2074

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