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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
14 Results for "
roflumilast
" in MedChemExpress (MCE) Product Catalog:
Products (14)
14 Results for "roflumilast" in MCE Product Catalog:
14
14 Publications Verification
Synonyms: APTA-2217; BYK 20869; B9302-107
Target:
Research Areas:
Roflumilast (APTA-2217) is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDE4A4, PDE4B1, and PDE4B2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells.
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1 Cited Publications
Research Areas:
Roflumilast N-oxide is a PDE type 4 inhibitor.
1
1 Cited Publications
Cat. No.: HY-15455S
CAS No.: 1398065-69-4
Synonyms: APTA-2217-d4; BYK 20869-d4; B9302-107-d4
Cat. No.: HY-100639R
CAS No.: 292135-78-5
Research Areas:
Roflumilast N-oxide (Standard) is the analytical standard of Roflumilast N-oxide. This product is intended for research and analytical applications. Roflumilast N-oxide is a PDE type 4 inhibitor.
Cat. No.: HY-100640
CAS No.: 1391052-76-8
Target:
Research Areas:
Roflumilast Impurity E is the impurity of Roflumilast. Roflumilast(Daliresp) is a agent which acts as a selective and long-acting inhibitor of the enzyme PDE-4 with an IC50 value of 0.8 nM.
Cat. No.: HY-15455R
CAS No.: 162401-32-3
Synonyms: APTA-2217 (Standard); BYK 20869 (Standard); B9302-107 (Standard)
Research Areas:
Roflumilast (Standard) is the analytical standard of Roflumilast. This product is intended for research and analytical applications. Roflumilast (APTA-2217) is a selective PDE4 inhibitor with IC50s of 0.7, 0.9, 0.7, and 0.2 nM for PDE4A1, PDEA4, PDEB1, and PDEB2, respectively, without affecting PDE1, PDE2, PDE3 or PDE5 isoenzymes from various cells.
Cat. No.: HY-100640R
CAS No.: 1391052-76-8
Research Areas:
Roflumilast Impurity E (Standard) is the analytical standard of Roflumilast Impurity E. This product is intended for research and analytical applications. Roflumilast Impurity E is the impurity of Roflumilast. Roflumilast(Daliresp) is a agent which acts as a selective and long-acting inhibitor of the enzyme PDE-4 with an IC50 value of 0.8 nM.
Cat. No.: HY-15455S2
CAS No.: 1189992-00-4
Synonyms: APTA-2217-d3; BYK 20869-d3; B9302-107-d3
Cat. No.: HY-168558
Target:
Research Areas:
PDE4B/D-IN-4 (compound 4p) is a potent inhibitor of PDE-4B and PDE-4D, with IC50s of 5.50 nM and 6.81 nM, respectively. PDE4B/D-IN-4 shows an increase in the level of intracellular cAMP .
Cat. No.: HY-W102746
CAS No.: 1391052-24-6
Synonyms: 3,4-Di(cyclopropylmethoxy) roflumilast
Target:
Research Areas:
Roflumilast impurity 1 (3,4-Di(cyclopropylmethoxy) roflumilast) is an impurity of Roflumilast.
Cat. No.: HY-W102745
CAS No.: 475271-62-6
Target:
Research Areas:
Roflumilast impurity 4 is an impurity of Roflumilast.
Cat. No.: HY-W1123449
CAS No.: 3031785-18-6
Target:
Research Areas:
Roflumilast impurity 3 is an impurity of Roflumilast.
Cat. No.: HY-Z18067
CAS No.: 1412448-29-3
Target:
Research Areas:
Roflumilast impurity 2 is an impurity of Roflumilast.
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