AChE-IN-81
AChE-IN-81 (compound 22) is a potent, irreversible and selective AChE inhibitor. AChE-IN-81 inhibits activity on AChE with inhibitory rates of 80.0%, with an IC50 of 3.7 μM. AChE-IN-81 binds to AChE with a binding affinity (Kd) of 5.37 μM. AChE-IN-81 effectively reduces in zebrafish brain cells. AChE-IN-81 exhibits potential neuroprotective activities on H2O2-induced SH-SY5Y cell injury model.
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- Formel: C37H54ClNO5
- Molecular Weight:628.28
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Help & FAQs
Biologische Aktivität
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AChE 3.7 μM (IC50) |
AChE 5.37 μM (Kd) |
Chemical Information
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Molecular Weight 628.28
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Formel C37H54ClNO5
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SMILES
ClC1=CC=CC=C1CNC([C@@]23CC[C@@]4(C)[C@]5(C)CC[C@@]6([H])[C@@](CO)(C)[C@@H](O)[C@H](O)C[C@]6(C)[C@@]5([H])CC=C4[C@@]([H])2[C@](C)(O)[C@H](C)CC3)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
AChE-IN-81 Related Classifications
HY-170925 Related Classifications
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