Pimavanserin-d4
Pimavanserin-d4 (ACP-103-d4) is the deuterium labeled Pimavanserin (HY-14557). Pimavanserin is a selective, brain-penetrant, inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- Formel: C25H30D4FN3O2
- Molecular Weight:431.58
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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Unlabeled Cas 706779-91-1
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Molecular Weight 431.58
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Formel C25H30D4FN3O2
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SMILES
CC(C)COC1=CC=C(CNC(N(CC2=C([2H])C([2H])=C(F)C([2H])=C2[2H])C3CCN(C)CC3)=O)C=C1
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Synonyms
ACP-103-d4
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)