ETP-45835
ETP-45835 is slective and potent MNK inhibitor with IC50s of 575 nM and 646 nM for MNK1 and MNK2, respectively. ETP-45835 shows little activity against 24 other kinases. ETP-45835 inhibits eIF4E Ser209 phosphorylation in cells, and has anticancer effects.
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- No. CAS: 794510-70-6
- Fòrmula: C13H16N4
- Peso molecular:228.29
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
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Help & FAQs
Actividad biológica
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MNK1 575 nM (IC50) |
MNK2 646 nM (IC50) |
Chemical Information
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No. CAS 794510-70-6
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Peso molecular 228.29
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Fòrmula C13H16N4
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SMILES
N=1C=CC(=CC1)C2=NNC(=C2)C3CCNCC3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
ETP-45835 Related Classifications
HY-W846144 Related Classifications
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