1. Signaling Pathways
  2. MAPK/ERK Pathway
  3. MNK
  4. MNK Inhibitors

MNK Inhibitors

MNK1

MNK2

MNK

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

MNK Inhibitors
Product Name MNK1 MNK2 MNK Purity
Tomivosertib
MNK1, IC50: 1-2 nM
MNK2, IC50: 1-2 nM
  99.92%
Tinodasertib
MNK1, IC50: 64 nM
MNK2, IC50: 86 nM
  99.69%
CGP 57380
MNK1, IC50: 2.2 μM
    98.0%
SLV-2436
MNK1, IC50: 10.8 nM
MNK2, IC50: 5.4 nM
  98.53%
ETC-168
MNK1, IC50: 23 nM
MNK2, IC50: 43 nM
 
Cercosporamide    
Mnk
≥98.0%
EB1
MNK1, IC50: 0.69 μM
MNK2, IC50: 9.4 μM
 
MNK inhibitor 9
MNK1, IC50: 0.003 μM
MNK2, IC50: 0.003 μM
 
MNK1/2-IN-6
MNK1, IC50: 2.3 nM
MNK2, IC50: 3.4 nM
 
K783-0308  
MNK2, IC50: 406 nM