NBI-75043
NBI-75043 is an antagonist of H1 receptor.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 873693-47-1
- Fòrmula: C19H22N2S
- Peso molecular:310.46
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Ver todos los productos específicos de isoformas Histamine Receptor
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Actividad biológica
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | IC50 |
5.3 μM
Compound: 2, (-)-R
|
Displacement of [3H]N-methylscopolamine from human muscarinic M1 receptor expressed in CHO Flp-In cells after 90 mins by scintillation counting
Displacement of [3H]N-methylscopolamine from human muscarinic M1 receptor expressed in CHO Flp-In cells after 90 mins by scintillation counting
|
[PMID: 20188547] |
| HEK293 | IC50 |
1.4 μM
Compound: 2a
|
Inhibition of human ERG expressed in HEK293 cells by patch-clamp technique
Inhibition of human ERG expressed in HEK293 cells by patch-clamp technique
|
[PMID: 19663387] |
Chemical Information
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No. CAS 873693-47-1
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Peso molecular 310.46
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Fòrmula C19H22N2S
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SMILES
CN(C)CCC1=C([C@H](C2=CC=CC=N2)C)C3=CC=CC=C3S1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)