Mazisotine
Based on 1 Customer Validation
Mazisotine (CNTX-0290) is an orally active, non-opioid somatostatin receptor 4 (SSTR4) agonist with an EC50 of 4.7 nM. Mazisotine exerts significant analgesic effects in various nociceptive (inflammatory, osteoarthritic) and neuropathic pain models. Mazisotine can be used for pain research.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 99.54%
- CAS 番号: 1638588-92-7
- 分子式: C16H23N3O2
- 分子量:289.37
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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Bioactive Compound Library Max
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MCE Bioactive Compound Library
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GPCR/G Protein Compound Library
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生物活性
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SSTR4 4.7 nM (EC50) |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 1638588-92-7
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性状 Solid
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分子量 289.37
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分子式 C16H23N3O2
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Color White to off-white
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SMILES
CC(C=CC=N1)=C1OCC(C)(C)NC([C@H]2[C@@]3([H])[C@]2([H])CNC3)=O
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別名
LY3556050; CNTX-0290
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 125 mg/mL (431.97 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (271 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.4558 mL | 17.2789 mL | 34.5578 mL | 86.3946 mL |
| 5 mM | 0.6912 mL | 3.4558 mL | 6.9116 mL | 17.2789 mL | |
| 10 mM | 0.3456 mL | 1.7279 mL | 3.4558 mL | 8.6395 mL | |
| 15 mM | 0.2304 mL | 1.1519 mL | 2.3039 mL | 5.7596 mL | |
| 20 mM | 0.1728 mL | 0.8639 mL | 1.7279 mL | 4.3197 mL | |
| 25 mM | 0.1382 mL | 0.6912 mL | 1.3823 mL | 3.4558 mL | |
| 30 mM | 0.1152 mL | 0.5760 mL | 1.1519 mL | 2.8798 mL | |
| 40 mM | 0.0864 mL | 0.4320 mL | 0.8639 mL | 2.1599 mL | |
| 50 mM | 0.0691 mL | 0.3456 mL | 0.6912 mL | 1.7279 mL | |
| 60 mM | 0.0576 mL | 0.2880 mL | 0.5760 mL | 1.4399 mL | |
| 80 mM | 0.0432 mL | 0.2160 mL | 0.4320 mL | 1.0799 mL | |
| 100 mM | 0.0346 mL | 0.1728 mL | 0.3456 mL | 0.8639 mL |
Mazisotine 関連分類
HY-139347 関連分類
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