1. Membrane Transporter/Ion Channel
  2. SGLT
  3. LX2761

LX2761 

Cat. No.: HY-101122
Handling Instructions

LX2761 is chemically stable and potent inhibitor against sodium-dependent glucose cotransporter 1 (SGLT1) and SGLT2 in vitro with IC50s of 2.2 nM and 2.7nM for hSGLT1 and hSGLT2, but displays specific SGLT1 inhibition in the gastrointestinal (GI) tract.

For research use only. We do not sell to patients.

LX2761 Chemical Structure

LX2761 Chemical Structure

CAS No. : 1610954-97-6

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Description

LX2761 is chemically stable and potent inhibitor against sodium-dependent glucose cotransporter 1 (SGLT1) and SGLT2 in vitro with IC50s of 2.2 nM and 2.7nM for hSGLT1 and hSGLT2, but displays specific SGLT1 inhibition in the gastrointestinal (GI) tract[1].

IC50 & Target

IC50: 2.2 nM (hSGLT1), 2.7nM (hSGLT2)[1]

Molecular Weight

601.80

Formula

C₃₂H₄₇N₃O₆S

CAS No.

1610954-97-6

SMILES

CC1=CC=C([[email protected]]2[[email protected]](O)[[email protected]@H](O)[[email protected]](O)[[email protected]@H](SC)O2)C=C1CC3=CC=C(CCCC(NC(C(NCCN(C)C)=O)(C)C)=O)C=C3

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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