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TA-0201

TA-0201 is a novel orally active, competitive, non-peptide endothelin receptor antagonist. TA-0201 antagonizes the specific binding of [125I]ET-1 to cloned human receptors of ETA and ETB with Ki values of 15 pM and 41 nM, respectively. TA-0201 inhibits the pressor response to the exogenous big ET-1.

For research use only. We do not sell to patients.

  • CAS No.: 169679-53-2
  • Formula: C27H28BrN5O5S
  • Molecular Weight:614.51
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • TA-0201 Chemical Structure
    TA-0201 Chemical Structure
CAS No.: 169679-53-2
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All Endothelin Receptor Isoforms

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  • TA-0201 Chemical Structure
    TA-0201 Chemical Structure
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  • TA-0201