1 Result for "

GSNOR-IN-1

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "GSNOR-IN-1" in MCE Product Catalog:

Cat. No.: HY-176712
Target:  

GSNOR Apoptosis

Research Areas:  

Neurological Disease

GSNOR-IN-1, a prodrug of GSNOR-IN-2 (HY-176275), is a BBB-penetrable S-nitrosoglutathione reductase (GSNOR) inhibitor. GSNOR-IN-1 has significant protective activity against OGD/R-induced injury. GSNOR-IN-1 regulates calcium signaling and synaptic function via Clstn1 S-nitrosation and inhibits neuronal apoptosis. GSNOR-IN-1 significantly reduces infarct volume while improving neurological deficits in ischemic stroke rat models. GSNOR-IN-1 has neuroprotective activity, promising for ischemic stroke research [1].
loading...
    loading...