15 Results for "

Ivabradine

" in MedChemExpress (MCE) Product Catalog:
Products (15)

15 Results for "Ivabradine" in MCE Product Catalog:

3
3 Cited Publications
Cat. No.: HY-B0162A
CAS No.: 148849-67-6
Ivabradine hydrochloride is a potent and orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits the cardiac pacemaker current (If). Ivabradine hydrochloride reduces dose-dependently heart rate without modification of blood pressure. Ivabradine hydrochloride shows anticonvulsant, anti-ischaemic and anti-anginal activity .
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3
3 Cited Publications
Cat. No.: HY-B0162
CAS No.: 155974-00-8
Target:  

HCN Channel

Research Areas:  

Cardiovascular Disease Cancer

Ivabradine is a potent and orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits the cardiac pacemaker current (If). Ivabradine reduces dose-dependently heart rate without modification of blood pressure. Ivabradine shows anticonvulsant, anti-ischaemic and anti-anginal activity .
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Cat. No.: HY-12778
CAS No.: 1246638-08-3
Purity:  99.63%
Synonyms: Ivabradine metabolite N-Demethyl Ivabradine hydrochloride
N-Demethyl Ivabradine (hydrochloride) is a metabolite of Ivabradine, which is a specific inhibitor of the funny channel.
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Cat. No.: HY-B0162AS
CAS No.: 2070009-63-9
Ivabradine-d6 hydrochloride is the deuterium labeled Ivabradine hydrochloride. Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent.
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Cat. No.: HY-B0162AS1
CAS No.: 1217809-61-4
Ivabradine-d3 (hydrochloride) is the deuterium labeled Ivabradine hydrochloride. Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent.
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Cat. No.: HY-12778R
CAS No.: 1246638-08-3
Synonyms: N-Demethyl Ivabradine hydrochloride (Standard)
Ivabradine metabolite N-Demethyl Ivabradine (hydrochloride) (Standard) is the analytical standard of Ivabradine metabolite N-Demethyl Ivabradine (hydrochloride). This product is intended for research and analytical applications. 0
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Cat. No.: HY-12778S
CAS No.: 2070009-60-6
Purity:  ≥98.0%
Synonyms: Ivabradine metabolite N-demethyl Ivabradine-d6 hydrochloride
N-Demethyl Ivabradine-d6 (hydrochloride) is the deuterium labeled N-Demethyl Ivabradine, which is a metabolite of Ivabradine.
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Cat. No.: HY-B0162AR
CAS No.: 148849-67-6
Ivabradine hydrochloride (Standard) is the analytical standard of Ivabradine hydrochloride. This product is intended for research and analytical applications. Ivabradine hydrochloride is a potent and orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits the cardiac pacemaker current (If). Ivabradine hydrochloride reduces dose-dependently heart rate without modification of blood pressure. Ivabradine hydrochloride shows anticonvulsant, anti-ischaemic and anti-anginal activity .
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Cat. No.: HY-B0162S
CAS No.: 2070009-62-8
Ivabradine-d6 is the deuterium labeled Ivabradine . Ivabradine is a potent and orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits the cardiac pacemaker current (If). Ivabradine reduces dose-dependently heart rate without modification of blood pressure. Ivabradine shows anticonvulsant, anti-ischaemic and anti-anginal activity .
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Cat. No.: HY-131283
CAS No.: 304464-97-9
Target:  

Drug Metabolite

Research Areas:  

Endocrinology

8-Demethyl Ivabradine is a metabolite of Ivabradine. Ivabradine is an orally bioavailable, hyperpolarization-activated, cyclic nucleotide-gated (HCN) channel blocker .
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Cat. No.: HY-131281
CAS No.: 1428869-91-3
Target:  

Drug Metabolite

Research Areas:  

Others

Ivabradine impurity 1 is an Ivabradine impurity. Ivabradine is an orally bioavailable, hyperpolarization-activated, cyclic nucleotide-gated (HCN) channel blocker .
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Cat. No.: HY-131282
CAS No.: 73954-34-4
Target:  

Drug Metabolite

Research Areas:  

Others

Ivabradine impurity 2 is an Ivabradine impurity. Ivabradine is an orally bioavailable, hyperpolarization-activated, cyclic nucleotide-gated (HCN) channel blocker .
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Cat. No.: HY-143970S
CAS No.: 2733718-12-0
Ivabradine impurity 7-d6 is the deuterium labeled Ivabradine impurity 7 .
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Cat. No.: HY-B0162B
CAS No.: 1202000-62-1
Ivabradine sulfate is a potent and orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits the cardiac pacemaker current (If). Ivabradine sulfate reduces dose-dependently heart rate without modification of blood pressure. Ivabradine sulfate shows anticonvulsant, anti-ischaemic and anti-anginal activity .
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Cat. No.: HY-100633S
CAS No.: 1346600-74-5
Synonyms: S-18982-d6 hydrochloride
N-Demethy Ivabradine-d6 (hydrochloride) is the deuterium labeled N-Demethy Ivabradine hydrochloride .
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