4 Results for "

YM09538

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "YM09538" in MCE Product Catalog:

Cat. No.: HY-106720
CAS No.: 85320-68-9
Purity:  98.69%
Synonyms: YM 09538
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Amosulalol (YM 09538) is an orally active and dual inhibitor of α1/β1-Adrenergic Receptor. Amosulalol exhibits antihypertensive activity via α1-Adrenergic Receptor inhibition. Amosulalol decreases reflexogenic increases in heart rate and plasma renin activity (PRA) via β1-Adrenergic Receptor inhibition in spontaneously hypertensive rats (SHR) .
loading...
    loading...
Cat. No.: HY-106720A
CAS No.: 70958-86-0
Synonyms: YM 09538 hydrochloride
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Amosulalol (YM 09538) hydrochloride is an orally active and dual inhibitor of α1/β1-Adrenergic Receptor. Amosulalol hydrochloride exhibits antihypertensive activity via α1-Adrenergic Receptor inhibition. Amosulalol hydrochloride decreases reflexogenic increases in heart rate and plasma renin activity (PRA) via β1-Adrenergic Receptor inhibition in spontaneously hypertensive rats (SHR) .
loading...
    loading...
Cat. No.: HY-106720B
CAS No.: 94666-15-6
Synonyms: (-)-YM 09538
Target:  

Adrenergic Receptor

Research Areas:  

Others

(-)-Amosulalol ((-)-YM 09538) is an isomer of Amosulalol (HY-106720), an orally active dual inhibitor of α1/β1-adrenergic receptors. Amosulalol exhibits antihypertensive activity by inhibiting α1-adrenergic receptors. Amosulalol reduces the reflex increase in heart rate and plasma renin activity (PRA) in spontaneously hypertensive rats (SHR) by inhibiting β1-adrenergic receptors.
loading...
    loading...
Cat. No.: HY-106720C
CAS No.: 94666-17-8
Synonyms: (+)-YM 09538
Target:  

Adrenergic Receptor

Research Areas:  

Others

(+)-Amosulalol ((+)-YM 09538) is an isomer of Amosulalol (HY-106720), an orally active dual inhibitor of α1/β1-adrenergic receptors. Amosulalol exhibits antihypertensive activity by inhibiting α1-adrenergic receptors. Amosulalol reduces the reflex increase in heart rate and plasma renin activity (PRA) in spontaneously hypertensive rats (SHR) by inhibiting β1-adrenergic receptors.
loading...
    loading...