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  2. TAK-448 acetate

TAK-448 acetate (Synonyms: MVT-602 (acetate))

Cat. No.: HY-P0076A Purity: 99.37%
Handling Instructions

TAK-448 acetate (MVT-602 acetate) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

TAK-448 acetate Chemical Structure

TAK-448 acetate Chemical Structure

CAS No. : 1470374-22-1

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 1273 In-stock
Estimated Time of Arrival: December 31
1 mg USD 150 In-stock
Estimated Time of Arrival: December 31
5 mg USD 450 In-stock
Estimated Time of Arrival: December 31
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50 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

TAK-448 acetate (MVT-602 acetate) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM[1].

IC50 & Target

IC50: 460 pM (KISS1R)[1]
EC50: 632 pM (KISS1R)[1]

In Vivo

TAK-448 acetate (0.01-3 mg/kg; given i.h.; dosings on day 0 and 28) has greater anti-tumor effects in VCaP xenograft model[2].

Animal Model: Rat VCaP xenograft androgen-sensitive prostate cancer model (7-week-old rats)
Dosage: 0.01, 0.03, 0.3, 3 mg/kg
Administration: Given i.h.; dosings on day 0 and 28
Result: Had greater anti-tumor effects in VCaP xenograft model.
Clinical Trial
Molecular Weight

1285.41

Formula

C₆₀H₈₄N₁₆O₁₆

CAS No.

1470374-22-1

Sequence

Ac-D-Tyr-D-Trp-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NH2

Sequence Shortening

Ac-Y-{Hyp}-NTFGLRW-NH2

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -80°C 2 years
  -20°C 1 year
In solvent -80°C 6 months
  -20°C 1 month
References
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TAK-448 acetate
Cat. No.:
HY-P0076A
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