1. GPCR/G Protein
  2. Somatostatin Receptor

SSTR5 antagonists 1 

Cat. No.: HY-102037
Handling Instructions

SSTR5 antagonists 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a)

For research use only. We do not sell to patients.

SSTR5 antagonists 1 Chemical Structure

SSTR5 antagonists 1 Chemical Structure

CAS No. : 1628741-91-2

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Description

SSTR5 antagonists 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a)[1]

IC50 & Target

IC50: 9.6 nM (hSSTR5), 57 nM (mSSTR5)[1]

References
Molecular Weight

511.59

Formula

C₂₈H₃₄FN₃O₅

CAS No.

1628741-91-2

SMILES

OC(C1CCN(C2=NOC3(CN(CC4=CC(OCC)=C(C5=CC=C(F)C=C5)C(OCC)=C4)C3)C2)CC1)=O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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Product Name:
SSTR5 antagonists 1
Cat. No.:
HY-102037
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SSTR5 antagonists 1

Cat. No.: HY-102037