YM218 free base
YM218 free base is an orally active non-peptide vasopressin (AVP) receptor antagonist. YM218 free base has a high affinity for rat liver V1A receptors with a Ki value of 0.50 nM; it has a lower affinity for rat pituitary V1B, kidney V2, and uterine oxytocin receptors with Ki values of 1510 nM, 72.2 nM, and 150 nM, respectively. YM218 free base can be used in the study of diabetes and kidney disease.
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- CAS. Nr.: 387816-81-1
- Formel: C35H38F2N4O4
- Molecular Weight:616.70
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Biologische Aktivität
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Rat liver V1a Receptor 0.5 nM (Ki) |
Rat pituitary V1b receptor 1510 nM (Ki) |
Rat kidney V2 receptor 72.2 nM (Ki) |
Chemical Information
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CAS. Nr. 387816-81-1
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Molecular Weight 616.70
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Formel C35H38F2N4O4
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SMILES
O=C(NC1=CC=C(C=C1)C(N2CCC(F)(/C(C3=CC=CC=C32)=C\C(N4CCC(CC4)N5CCCCC5)=O)F)=O)C6=C(OC=C6)C
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
YM218 free base Related Classifications
HY-118918 Related Classifications
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