1. Signaling Pathways
  2. GPCR/G Protein
  3. Vasopressin Receptor
  4. Vasopressin Receptor Inhibitors

Vasopressin Receptor Inhibitors

V1a Receptor 

V1b Receptor 

V2 Receptor 

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Vasopressin Receptor Inhibitors, Agonists, Antagonists, Activators & Ligands
Product Name V1a Receptor  V1b Receptor  V2 Receptor  Purity
Tolvaptan    
V2 Receptor 
99.95%
Argipressin    
V2 Receptor 
98.71%
Conivaptan hydrochloride    
V2 Receptor 
99.95%
SR 49059
V1a Receptor 
    99.33%
AGN-190851    
V2 Receptor 
Terlipressin diacetate  
V1b Receptor 
  98.86%
Mozavaptan    
V2 Receptor 
99.71%
Balovaptan
V1a Receptor 
    99.89%
D[LEU4,LYS8]-VP TFA  
V1b Receptor 
  98.97%
Lixivaptan    
V2 Receptor 
99.67%
Mozavaptan hydrochloride    
V2 Receptor 
99.80%
SRX246
V1a Receptor 
    99.76%
Fedovapagon    
V2 Receptor , EC50: 24 nM
99.43%
TC OT 39
Avprla vasopressin receptor, Ki: 300 nM
   
RG7713
V1a Receptor 
    99.92%
Vasopressin Dimer (parallel) TFA    
V2 Receptor 
99.55%
Vasopressin V2 receptor antagonist 1    
V2 Receptor , Ki: 3.8 nM
V1a/V2 antagonist 1
human V1a Receptor, Ki: 0.13 nM
human V1a Receptor, IC50: 2.2 nM
 
human V2 Receptor, Ki: 0.53 nM
Vasopressin Dimer (anti-parallel) TFA    
V2 Receptor 
VA-111913
V1a Receptor , Ki: 1.74 nM
   
XYDC2050    
V2 Receptor , IC50: 27 nM
V2 Receptor , Ki: 2.8 nM
V1b Receptor antagonist-1  
V1b Receptor 
 
Mozavaptan-d6    
V2 Receptor 
ML389
V1a Receptor 
   
Pecavaptan
human V1a Receptor, IC50: 3.6 nM
canine V1a Receptor, IC50: 4.4 nM
 
human V2 Receptor, IC50: 1.7 nM
canine V2 Receptor, IC50: 1.3 nM
Conivaptan    
V2 Receptor 
L-364918    
V2 Receptor , Ki: 2400 nM
YM218 free base
Rat liver V1a Receptor, Ki: 0.5 nM
Rat pituitary V1b receptor, Ki: 1510 nM
Rat kidney V2 receptor, Ki: 72.2 nM
DM-4111    
V2 Receptor 
Tolvaptan-d7    
V2 Receptor 
TASP0434299  
V1b Receptor