Bromodomain inhibitor-9
Bromodomain inhibitor-9 is a Bromodomains inhibitor that selectively inhibits BRD4-1 (Kd: 12 nM). Bromodomain inhibitor-9 can be used in the research of diseases or conditions associated with systemic or tissue inflammation, lipid metabolism, fibrosis or chronic autoimmune diseases.
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- CAS No.: 1870849-34-5
- Formule: C24H28N4O5S
- Masse moléculaire:484.57
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
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BRD4-1 12 nM (Kd) |
BRD4-2 5600 nM (Kd) |
Bromodomain inhibitor-9 (Compound 99, 1 h) inhibits LPS induced cytokines (IL12P40) release in PBMCs, with an IC50 value of 400 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1870849-34-5
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Masse moléculaire 484.57
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Formule C24H28N4O5S
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SMILES
O=C1C=C(C)C2=C(N1)C=C(C)C(NC(C3=CC(S(=O)(N(C)C)=O)=CC=C3N4CCOCC4)=O)=C2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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