Mayumbine
Mayumbine (19-Epiajmalicine) is a natural alkaloid.
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- CAS No.: 25532-45-0
- Formule: C21H24N2O3
- Masse moléculaire:352.43
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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D2 Receptor 3.5 μM (IC50) |
A1AR 320 nM (IC50) |
Mayumbine competitively inhibits the binding of 3H-flunitrazepam to GABAA/BZD receptors in rat cerebral cortex, hippocampus, and cerebellar membrane preparations, reducing binding affinity (Kd) but not altering the maximum number of binding sites (Bmax), and was identified as a partial agonist[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 25532-45-0
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Masse moléculaire 352.43
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Formule C21H24N2O3
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SMILES
COC(C1=CO[C@@H]([C@@]2([C@@]1(C[C@]3(C4=C(C5=C(N4)C=CC=C5)CCN3C2)[H])[H])[H])C)=O
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Synonyms
19-Epiajmalicine
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Structure Classification
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Initial Source
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)