(+)-Alprenolol
(+)-Alprenolol ((R)-Alprenolol; D-Alprenolol) is a 5-HT1A receptor antagonist with a Ki value of 5400 nM. (+)-Alprenolol also acts as a non-selective β-receptor (β-receptor) blocker. (+)-Alprenolol can be used in the research of cardiovascular and cerebrovascular diseases.
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- CAS. Nr.: 23846-72-2
- Formel: C15H23NO2
- Molecular Weight:249.35
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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5-HT1A Receptor 5400 nM (Ki) |
β-adrenoceptor |
(+)-Alprenolol ((R)-5) binds to the human 5-HT1A Asn386Val mutant receptor with a Ki of 56000 nM, showing 10-fold lower affinity than for the wild-type receptor and reduced stereoselectivity relative to its S enantiomer[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS. Nr. 23846-72-2
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Molecular Weight 249.35
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Formel C15H23NO2
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SMILES
O(C[C@@H](CNC(C)C)O)C1=C(CC=C)C=CC=C1
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Synonyms
(R)-Alprenolol; D-Alprenolol
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
(+)-Alprenolol Related Classifications
HY-165357 Related Classifications
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