BChE-IN-20
BChE-IN-20 (compound 7c) is a highly potent BChE-selective inhibitor and exhibits IC50s of 105 and 2.3 nM for eqBChE and hBChE, respectively. BChE-IN-20 inhibits P glycoprotein with IC50 of 0.27 μM. BChE-IN-20 is a promising template to improve design and development of BChE-selective ligands of pharmaceutical interest, including inhibitors and fluorogenic probes.
For research use only. We do not sell to patients.
- CAS No.: 1428439-79-5
- Formula: C27H39N5O2
- Molecular Weight:465.63
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 1428439-79-5
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Molecular Weight 465.63
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Formula C27H39N5O2
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SMILES
O=C(OC)/C(C1)=C/N(C(C)C)CCC2=C1C(NCCCN(CC)CC)=NC(C3=CC=CC=C3)=N2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)