VUF14480
VUF14480 is a partial agonist of histamine H4 (hH4) receptor-mediated G protein signalling and β-arrestin2 recruitment. VUF14480 binds covalently to hH4 receptor (pKi: 6.3 for hH4-WT receptor). VUF14480 partially induces hH4 receptor-mediated G protein activation and β-arrestin2 recruitment. VUF14480 can be used in the research of inflammatory diseases.
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- No. CAS: 1605304-31-1
- Fòrmula: C17H20N4
- Peso molecular:280.38
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
pKi: 6.3 for hH4-WT receptor[1]
Chemical Information
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No. CAS 1605304-31-1
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Peso molecular 280.38
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Fòrmula C17H20N4
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SMILES
N=1C(=NC(=CC1C=2C=CC=CC2)N3CCN(C)CC3)C=C
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)