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Cat. No.: HY-119768

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(±)-BAK2-66

(±)-BAK2-66 is a selectivity dopamine D3 receptor antagonist with theK_i values of 1nM and 960 nM for D3R and D2R, respectively. (±)-BAK2-66 can be used for study in animal models of addiction.

For research use only. We do not sell to patients.

CAS No.: 1301178-83-5
Formula: C₂₃H₂₄Cl₂FN₃O₂
Molecular Weight:464.36

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (264 KB)

(±)-BAK2-66 Chemical Structure

CAS No.: 1301178-83-5

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

(±)-BAK2-66 is a selectivity dopamine D3 receptor antagonist with theK_i values of 1nM and 960 nM for D3R and D2R, respectively. (±)-BAK2-66 can be used for study in animal models of addiction^[1].

All Dopamine Receptor Isoforms :

Chemical Information

CAS No. 1301178-83-5
Molecular Weight 464.36
Formula C₂₃H₂₄Cl₂FN₃O₂
SMILES

O=C(NCCC(CN1CCN(CC1)C2=CC=CC(Cl)=C2Cl)F)C3=CC4=CC=CC=C4O3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (264 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Kumar V, et al. Chiral Resolution and Serendipitous Fluorination Reaction for the Selective Dopamine D3 Receptor Antagonist BAK2-66. ACS Med Chem Lett. 2014;5(6):647-651. Published 2014 Mar 24. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Biological Activity
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Chemical Information
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References

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(±)-BAK2-66

All Dopamine Receptor Isoforms