1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
  3. Odapipam

Odapipam (Synonyms: NNC 756)

Cat. No.: HY-129059
Handling Instructions

Odapipam (NNC 756) is a selective, high affinity and benzazepine dopamine D1 receptor antagonist with a Kd of 0.18 nM. Odapipam is also a superior positron emission tomography (PET) radiotracer.

For research use only. We do not sell to patients.

Odapipam Chemical Structure

Odapipam Chemical Structure

CAS No. : 131796-63-9

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Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Description

Odapipam (NNC 756) is a selective, high affinity and benzazepine dopamine D1 receptor antagonist with a Kd of 0.18 nM. Odapipam is also a superior positron emission tomography (PET) radiotracer[1][2].

IC50 & Target

Dopamine D1 receptor[1]

In Vivo

The metabolism of Odapipam has been studied with phenobarbital-induced rat liver microsomes. During the incubation of Odapipam, five different metabolites are formed. The electron-ionization (EI+) mass spectra of the metabolites indicated the formation of N-desmethyl-Odapipam, 1-hydroxy-Odapipam, the two isomers of 3′-hydroxy-Odapipam and a metabolite which is dehydrogenated in the dihydrobenzofuran moiety[3].

Molecular Weight

329.82

Formula

C₁₉H₂₀ClNO₂

CAS No.

131796-63-9

SMILES

OC1=C(Cl)C=C2CCN(C)C[[email protected]](C3=C(OCC4)C4=CC=C3)C2=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

OdapipamNNC 756NNC756NNC-756Dopamine ReceptorInhibitorinhibitorinhibit

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Odapipam
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