9 Results for "

Benzamide-d5

" in MedChemExpress (MCE) Product Catalog:
Products (9)

9 Results for "Benzamide-d5" in MCE Product Catalog:

1
1 Cited Publications
Referencia número: HY-P1103
No. CAS: 1030384-98-5
Target:  

CXCR

Áreas de investigación:  

Cancer

CTCE-9908 is a potent and selective CXCR4 antagonist. CTCE-9908 induces mitotic catastrophe, cytotoxicity and inhibits migration in CXCR4-expressing ovarian cancer cells .
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Referencia número: HY-P4070
No. CAS: 1188379-43-2
Target:  

Insulin Receptor

Áreas de investigación:  

Metabolic Disease

Insulin icodec is an Insulin (HY-P0035) analog that strongly but reversibly binds to albumin. Insulin icodec has long plasma half-life. Insulin icodec modulates insulin receptor activity, controls blood glucose levels, reduces HbA1c levels, and binds reversibly to human serum albumin. Insulin icodec can be used for the research of type 2 diabetes mellitus .
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Referencia número: HY-W711852
No. CAS: 1235489-47-0
Synonyms: Benzenecarboxamide-d5; Phenylamide-d5
Benzamide-d5 (Benzenecarboxamide-d5) is deuterium labeled Benzamide. Benzamide (Benzenecarboxamide) is a potent poly(ADP-ribose) polymerase (PARP) inhibitor. Benzamide has protective activity against both glutamate- and methamphetamine (METH)-induced neurotoxicity in vitro. Benzamide can attenuate the METH-induced dopamine depletions and exhibits neuroprotective activity in mice, also has no acute effect on striatal dopamine metabolism and does not reduce body temperature .
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Referencia número: HY-P1103A
Target:  

CXCR

Áreas de investigación:  

Cancer

CTCE-9908 TFA is a potent and selective CXCR4 antagonist. CTCE-9908 TFA induces mitotic catastrophe, cytotoxicity and inhibits migration in CXCR4-expressing ovarian cancer cells .
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Referencia número: HY-P11293
No. CAS: 1309855-53-5
Target:  

Melanocortin Receptor

Áreas de investigación:  

Cancer

DOTA-GGNle-CycMSHhex is a melanocortin-1 receptor (MC1R)-targeting peptide that can be radionuclide-labeled for melanoma imaging .
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Referencia número: HY-P4757
No. CAS: 108081-77-2
Target:  

Parasite

Áreas de investigación:  

Others

N1-Glutathionyl-spermidine disulfide is a substrate of trypanothione reductase .
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Referencia número: HY-P1321
No. CAS: 158859-98-4
Synonyms: 1229U91; GW1229
Áreas de investigación:  

Neurological Disease

GR231118, an analogue of the C-terminus of neuropeptide Y, is a potent , competitive and relative seletive antagonist at human neuropeptide Y Y receptor with a pKi of 10.4. GR231118 a potent agonist at the human neuropeptide Y Y4 receptor (pEC50=8.6; pKi=9.6) and a weak agonist at the human and rat neuropeptide YY2 and Y5 receptors. GR231118 also has high affinity for the mouse neuropeptide Y Y6 receptor (pKi= 8.8) .
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Referencia número: HY-P1321A
Synonyms: 1229U91 TFA; GW1229 TFA
Áreas de investigación:  

Neurological Disease

GR231118 TFA, an analogue of the C-terminus of neuropeptide Y, is a potent , competitive and relative seletive antagonist at human neuropeptide YY receptor with a pKi of 10.4. GR231118 a potent agonist at the human neuropeptide YY4 receptor (pEC50=8.6; pKi=9.6) and a weak agonist at the human and rat neuropeptide Y Y2 and Y5 receptors. GR231118 also has high affinity for the mouse neuropeptide YY6 receptor (pKi= 8.8) .
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Referencia número: HY-P11480
No. CAS: 3105660-96-3
Target:  

Trk Receptor

Áreas de investigación:  

Neurological Disease

TrkA/NGF-IN-1 (Peptide 19) is an inhibitor of protein-protein interactions between TrkA and NGF (IC50: 21 nM for human TrkA in PathHunter assay). TrkA/NGF-IN-1 shows an analgesic effect in a rat incisional pain model .
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