2 Results for "

JZY3032

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "JZY3032" in MCE Product Catalog:

Cat. No.: HY-184124
Research Areas:  

Cancer

JYZ3032 is an orally active super inhibitor of androgen receptor (AR) and p300/CBP. JYZ3032 redirects the catalytic activity of p300 and locks the complex in a transcriptionally inactive state, thereby inhibiting AR-driven transcription and proliferation. JYZ3032 induces deep and durable tumor regression in castration-resistant and patient-derived xenograft models, and exhibits good tolerability. JYZ3032 can be used in research related to metastatic castration-resistant prostate cancer and prostate cancer .
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Cat. No.: HY-184126
Target:  

Androgen Receptor

Research Areas:  

Cancer

JZY3221 is an androgen receptor (AR) inhibitor. JZY3221 binds to the AR ligand-binding domain to inhibit AR function. JZY3221 constitutes the AR inhibitory moiety of DALTAC JZY3032 (HY-184124). JZY3221 is applicable to research related to prostate cancer .
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