1 Result for "

PF07328948

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "PF07328948" in MCE Product Catalog:

Cat. No.: HY-159648
CAS No.: 2936625-34-0
Target:  

Endogenous Metabolite

Research Areas:  

Cardiovascular Disease

PF-07328948 is an orally effective BDK (branch chain ketoacid dehydrogenase kinase) inhibitor, with IC50 of 110 nM. PF-07328948 acts as a BCKDH (branch chain ketoacid dehydrogenase) enzyme complex degrader to enhance BCAA (branch chain amino acid) catabolism. PF-07328948 improves metabolic and heart failure end points in rats .
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