1 Result for "

chiauranib

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "chiauranib" in MCE Product Catalog:

Cat. No.: HY-124526
CAS No.: 1256349-48-0
Purity:  99.28%
Synonyms: Ibcasertib; CS2164
Research Areas:  

Cancer

Chiauranib (CS2164) is an orally active multi-target inhibitor against tumor angiogenesis. Chiauranib potently inhibits the angiogenesis-related kinases (VEGFR1, VEGFR2, VEGFR3, PDGFRα and c-Kit), mitosis-related kinase Aurora B, and chronic inflammation-related kinase CSF-1R, with IC50 values ranging from 1-9 nM. Chiauranib has strongly anticancer effects .