1. GPCR/G Protein
  2. Glucagon Receptor
  3. VU0453379

VU0453379 

Cat. No.: HY-116819
Handling Instructions

VU0453379 is a highly selective and central nervous system (CNS) penetrant positive allosteric modulator (PAM) of glucagon-like peptide-1R (GLP-1R) with an EC50 of 1.3 μM.

For research use only. We do not sell to patients.

VU0453379 Chemical Structure

VU0453379 Chemical Structure

CAS No. : 1638646-27-1

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Description

VU0453379 is a highly selective and central nervous system (CNS) penetrant positive allosteric modulator (PAM) of glucagon-like peptide-1R (GLP-1R) with an EC50 of 1.3 μM[1].

IC50 & Target

EC50: 1.3 μM (GLP-1R)[1]

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
Molecular Weight

434.57

Formula

C₂₆H₃₄N₄O₂

CAS No.

1638646-27-1

SMILES

O=C(NC[[email protected]]1N(CCC1)C(C)C)C(C2=C3N(C4=C2C=CC=C4)C)=CN(C3=O)C5CCCC5

Shipping

Room temperature in continental US; may vary elsewhere

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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VU0453379
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HY-116819
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VU0453379

Cat. No.: HY-116819