16 Results for "

Promethazine hydrochloride

" in MedChemExpress (MCE) Product Catalog:
Products (16)

16 Results for "Promethazine hydrochloride" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-B0781
CAS No.: 58-33-3
Promethazine hydrochloride is an orally active phenothiazine derivative with antihistaminic (H1), sedative, antiemetic, anticholinergic, and antimotion sickness properties. Promethazine hydrochloride is a potent H1 receptor antagonist and a mAChR antagonist. It also has a certain affinity for 5-HT2A and 5-HT2C receptors .
1
1 Cited Publications
Cat. No.: HY-B1296
CAS No.: 60-87-7
Synonyms: (±)-Promethazine
Target:  

Histamine Receptor

Research Areas:  

Neurological Disease

Promethazine is an orally active histamine receptor antagonist . Promethazine is first-generation antihistamine of the phenothiazine family, shows strong sedative and weak antipsychotic effects .
Cat. No.: HY-B0781S
CAS No.: 1173018-74-0
Promethazine-d4 (hydrochloride) is the deuterium labeled Promethazine hydrochloride. Promethazine hydrochloride is the first-generation antihistamine; strong antagonist of the H1 receptor and moderate mACh receptor antagonist, moderate affinity for 5-HT2A, 5-HT2C, D2 and α1-adrenergic receptors.
Cat. No.: HY-B1296S
CAS No.: 1189947-02-1
Synonyms: (±)-Promethazine-d6 hydrochloride
Promethazine-d6 (hydrochloride) is the deuterium labeled Promethazine hydrochloride. Promethazine hydrochloride is an orally active histamine receptor antagonist .
Cat. No.: HY-168958
CAS No.: 2247525-20-6
Research Areas:  

Cancer

Ferroptosis-IN-18 (51), a promethazine derivative, shows strong anti-ferroptosis and anti-oxidant properties. Ferroptosis-IN-18 (51) can be used in the research for intracerebral hemorrhage (ICH) .
Cat. No.: HY-Z9101
CAS No.: 7640-51-9
Target:  

Histamine Receptor

Research Areas:  

Neurological Disease

Promethazine sulfoxide is a metabolite of the histamine H1 receptor antagonist Promethazine (HY-B1296). It is formed from promethazine by the cytochrome P450 (CYP) isoform CYP2D6.
Cat. No.: HY-U00267
CAS No.: 4320-13-2
Target:  

Cholinesterase (ChE)

Research Areas:  

Inflammation/Immunology

Thiazinamium (chloride) possesses potent anticholinergic and antiallergic activity and inhibits TxB2 synthesis with IC50 value of 0.2 µM. Thiazinamium (chloride) is structurally similar to H-1 antagonists Promethazine (HY-B1296). Thiazinamium (chloride) stimulates the phosphatidylcholine secretion in adult rat type II pneumocytes .
Cat. No.: HY-B0781S1
Promethazine-d3 (hydrochloride) is deuterium labeled Promethazine (hydrochloride). Promethazine hydrochloride is an orally active phenothiazine derivative with antihistaminic (H1), sedative, antiemetic, anticholinergic, and antimotion sickness properties. Promethazine hydrochloride is a potent H1 receptor antagonist and a mAChR antagonist. It also has a certain affinity for 5-HT2A and 5-HT2C receptors .
Cat. No.: HY-B0781R
CAS No.: 58-33-3
Promethazine (hydrochloride) (Standard) is the analytical standard of Promethazine (hydrochloride). This product is intended for research and analytical applications. Promethazine hydrochloride is an orally active phenothiazine derivative with antihistaminic (H1), sedative, antiemetic, anticholinergic, and antimotion sickness properties. Promethazine hydrochloride is a potent H1 receptor antagonist and a mAChR antagonist. It also has a certain affinity for 5-HT2A and 5-HT2C receptors .
Cat. No.: HY-141739S
CAS No.: 1189892-93-0
Promethazine sulfoxide-d6 is the deuterium labeled Promethazine sulfoxide .
Cat. No.: HY-B1296S1
CAS No.: 1173147-64-2
Synonyms: (±)-Promethazine-d4; N,N-dimethyl-1-phenothiazin-10-yl-propan-2-amine-d4
Promethazine-d4 is a deuterated-labeled promethazine (HY-B0781). Promethazine is an orally active H1 receptor and mAChR antagonist with antihistamine (H1), sedative, antiemetic, anticholinergic, and anti-motion sickness properties .
Cat. No.: HY-Z9100
CAS No.: 60113-77-1
Target:  

Antibiotic

Research Areas:  

Infection

N-demethyl Promethazine hydrochloride is a metabolite of Phenothiazine (HY-Y0055). Phenothiazine is an antibiotic which has insecticidal, fungicidal, antibacterial and anthelmintic activities.
Cat. No.: HY-Z9099
CAS No.: 5568-90-1
Target:  

Drug Intermediate

Research Areas:  

Neurological Disease

Isopromethazine hydrochloride is an impurity in the pharmaceutical preparations of Promethazine (HY-B1296). Promethazine is an N-substituted phenothiazine with the actions and the uses of the antihistamines (H1-receptor antagonists) .
Cat. No.: HY-B1296R
CAS No.: 60-87-7
Synonyms: (±)-Promethazine (Standard)
Promethazine (Standard) is the analytical standard of Promethazine. This product is intended for research and analytical applications. Promethazine is an orally active histamine receptor antagonist . Promethazine is first-generation antihistamine of the phenothiazine family, shows strong sedative and weak antipsychotic effects .
Cat. No.: HY-B1296B
CAS No.: 67253-23-0
Target:  

Drug Isomer

Research Areas:  

Others

(R)-Promethazine is the R-enantiomer of Promethazine (HY-B1296). Promethazine is an orally active histamine receptor antagonist. Promethazine is first-generation antihistamine of the phenothiazine family, shows strong sedative and weak antipsychotic effects .
Cat. No.: HY-141742S
CAS No.: 1330173-19-7
N-Demethyl Promethazine-d3 (hydrochloride) is the deuterium labeled N-Demethyl Promethazine hydrochloride .
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