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Barbadin 

Cat. No.: HY-119706
Handling Instructions

Barbadin is a novel and selective β-arrestin/β2-adaptin interaction inhibitor, has IC50 values of 19.1 μM for β-arrestin1 and 15.6 μM for β-arrestin2. Barbadin blocks agonist-promoted endocytosis of the prototypical β2-adrenergic, V2-vasopressin and angiotensin-II type-1 receptors.

For research use only. We do not sell to patients.

Barbadin Chemical Structure

Barbadin Chemical Structure

CAS No. : 356568-70-2

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Description

Barbadin is a novel and selective β-arrestin/β2-adaptin interaction inhibitor, has IC50 values of 19.1 μM for β-arrestin1 and 15.6 μM for β-arrestin2. Barbadin blocks agonist-promoted endocytosis of the prototypical β2-adrenergic, V2-vasopressin and angiotensin-II type-1 receptors[1].

IC50 & Target

IC50: 19.1 μM (β-arrestin1); 15.6 μM (β-arrestin2)[1]

Molecular Weight

333.41

Formula

C₁₉H₁₅N₃OS

CAS No.

356568-70-2

SMILES

O=C1C(C(C2=CC=C(CC3=CC=CC=C3)C=C2)=CS4)=C4N=CN1N

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Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Barbadin
Cat. No.:
HY-119706
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