1. Signaling Pathways
  2. GPCR/G Protein
  3. Arrestin
  4. Arrestin Inhibitors

Arrestin Inhibitors

Arrestin-2/β-Arrestin 1

Arrestin-3/β-Arrestin 2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Arrestin Inhibitors, Agonists, Activators, Modulators & Inducers
Product Name Arrestin-2/β-Arrestin 1 Arrestin-3/β-Arrestin 2 Purity
Barbadin  
Arrestin-3/β-Arrestin 2
98.93%
TRV0109101
Arrestin-2/β-Arrestin 1
 
TRV-120027
Arrestin-2/β-Arrestin 1
  98.21%
IHCH-7086  
Arrestin-3/β-Arrestin 2
98.96%
DOR agonist 3  
Arrestin-3/β-Arrestin 2
5-HT2AR ligand 1  
Arrestin-3/β-Arrestin 2
GEP44  
Arrestin-3/β-Arrestin 2
B-007
Arrestin-2/β-Arrestin 1
Arrestin-3/β-Arrestin 2
ID110460002  
Arrestin-3/β-Arrestin 2
GPR183 inverse agonist-1  
Arrestin-3/β-Arrestin 2
Arrestin-3 modulator-1  
Arrestin-3/β-Arrestin 2
SLW131  
Arrestin-3/β-Arrestin 2, IC50: 6.0 μM
ID110460001
Arrestin-2/β-Arrestin 1
 
BMS-986331
Arrestin-2/β-Arrestin 1
Arrestin-3/β-Arrestin 2