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Cat. No.: HY-P1018

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IRL 1038

IRL 1038 is an endothelin B receptor selective antagonist with a K_i of 6-11 nM.

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CAS No.: 144602-02-8
Formule: C₆₈H₉₂N₁₄O₁₅S₂
Masse moléculaire:1409.67

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Please store the product under the recommended conditions in the Certificate of Analysis.

IRL 1038 Chemical Structure

CAS No.: 144602-02-8

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

IRL 1038 is an endothelin B receptor selective antagonist with a K_i of 6-11 nM^[1].

IC₅₀ & Target

Ki: 6-11 nM (endothelin B receptors), 0.4-0.7 μM (endothelin A receptors)^[1]

Voir tous les produits spécifiques à Isoform Endothelin Receptor :

ET_A
ET_B

Chemical Information

CAS No. 144602-02-8
Masse moléculaire 1409.67
Formule C₆₈H₉₂N₁₄O₁₅S₂
Sequence

Cys-Val-Tyr-Phe-Cys-His-Leu-Asp-Ile-Ile-Trp (Disulfide bridge:Cys1-Cys5)
Sequence Shortening

CVYFCHLDIIW (Disulfide bridge:Cys1-Cys5)
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (259 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Urade Y, et al. An endothelin B receptor-selective antagonist: IRL 1038, [Cys11-Cys15]-endothelin-1(11-21). FEBS Lett. 1992 Oct 12;311(1):12-6. doi: 10.1016/0014-5793(92)81355-p. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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IRL 1038

Voir tous les produits spécifiques à Isoform Endothelin Receptor

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

IRL 1038 Related Classifications

HY-P1018 Related Classifications