MK-8318
MK-8318 is a potent and selective CRTh2 receptor antagonist with a Ki of 5.0 nM.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 1416581-40-2
- Fòrmula: C27H26F4N2O5
- Peso molecular:534.50
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
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Actividad biológica
|
DP 5.0 nM (Ki) |
β-arrestin 3.5 nM (IC50) |
cAMP 8.0 nM (IC50) |
CYP3A4 50 μM (IC50) |
CYP2C9 50 μM (IC50) |
CYP2D6 50 μM (IC50) |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 1416581-40-2
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Peso molecular 534.50
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Fòrmula C27H26F4N2O5
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SMILES
FC1=CC=C(N(C(C2=CC=C(OC(F)(F)F)C=C2)=O)[C@@H](CCC3)[C@@H]3[C@H]4N(C(CCC(O)=O)=O)C5CC5)C4=C1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MK-8318 Related Classifications
HY-112604 Related Classifications
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