1. Membrane Transporter/Ion Channel
  2. Sodium Channel
  3. GX-201


Cat. No.: HY-131870
Handling Instructions

GX-201 is a selective NaV1.7 inhibitor, with an IC50 of <3.2 nM for hNaV1.7.

For research use only. We do not sell to patients.

GX-201 Chemical Structure

GX-201 Chemical Structure

CAS No. : 1788071-27-1

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GX-201 is a selective NaV1.7 inhibitor, with an IC50 of <3.2 nM for hNaV1.7[1].

In Vivo

GX-201 has a relatively long half-life in mice[1].
GX-201 produces analgesia at a free plasma concentration about 3 times the IC50 for high-affinity channel block[1].
GX-201 inhibits nociceptive responses induced by formalin and inflammatory pain caused by complete Freund’s adjuvant (CFA)[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Wild-Type Mice[1].
Dosage: 0.3, 1, 3 mg/kg.
Administration: Orally, once.
Result: Produced a dose-dependent inhibition of the nociceptive events.
Molecular Weight





Room temperature in continental US; may vary elsewhere.


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