DG013A formate
Based on 1 Customer Validation
DG013A (formate) is a phosphinic acid tripeptide mimetic inhibitor. DG013A (formate) displays significantly weak affinity for both ERAP1 (IC50=33 nM) and ERAP2 (IC50=11 nM). DG013A (formate) can be used for the research of autoimmune disease and cancer.
For research use only. We do not sell to patients.
- Purity: 99.57%
- Formula: C30H43N4O10P
- Molecular Weight:650.66
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Storage:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
Chemical Information
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Appearance Solid
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Molecular Weight 650.66
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Formula C30H43N4O10P
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Color White to off-white
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SMILES
O=P([C@@H](N)CCC1=CC=CC=C1)(O)C[C@@H](CC(C)C)C(N[C@H](C(N)=O)CC2=CNC3=CC=CC=C23)=O.O=CO.O=CO.O=CO
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 50 mg/mL (76.85 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
H2O : < 0.1 mg/mL (insoluble)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (272 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.5369 mL | 7.6845 mL | 15.3690 mL | 38.4225 mL |
| 5 mM | 0.3074 mL | 1.5369 mL | 3.0738 mL | 7.6845 mL | |
| 10 mM | 0.1537 mL | 0.7685 mL | 1.5369 mL | 3.8423 mL | |
| 15 mM | 0.1025 mL | 0.5123 mL | 1.0246 mL | 2.5615 mL | |
| 20 mM | 0.0768 mL | 0.3842 mL | 0.7685 mL | 1.9211 mL | |
| 25 mM | 0.0615 mL | 0.3074 mL | 0.6148 mL | 1.5369 mL | |
| 30 mM | 0.0512 mL | 0.2562 mL | 0.5123 mL | 1.2808 mL | |
| 40 mM | 0.0384 mL | 0.1921 mL | 0.3842 mL | 0.9606 mL | |
| 50 mM | 0.0307 mL | 0.1537 mL | 0.3074 mL | 0.7685 mL | |
| 60 mM | 0.0256 mL | 0.1281 mL | 0.2562 mL | 0.6404 mL |