DG013B formate

Cat. No.: HY-139907C: Data Sheet
SDS
Handling Instructions
FAQs
Technical Support

DG013B formate is an epimer of DG013A (HY-139907). DG013B formate has weak affinity for ERAP1 and ERAP2 and is often used as a negative control to study the binding properties of DG013A and its analogues to ERAP1 and ERAP2.

For research use only. We do not sell to patients.

DG013B formate Chemical Structure

Size	Stock	Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO ready for reconstitution	In-stock	Estimated Time of Arrival: December 31
Solution
10 mM * 1 mL in DMSO	In-stock	Estimated Time of Arrival: December 31
Solid
1 mg	In-stock	Estimated Time of Arrival: December 31
5 mg	In-stock	Estimated Time of Arrival: December 31
10 mg	In-stock	Estimated Time of Arrival: December 31
25 mg	In-stock	Estimated Time of Arrival: December 31
50 mg	Get quote
100 mg	Get quote

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This product is a controlled substance and not for sale in your territory.

Other Forms of DG013B formate:

DG013A formate In-stock
DG013A Get quote
DG013B Get quote

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Biological Activity
Purity & Documentation
References
Customer Review

Description

Molecular Weight

530.99

Formula

C₂₇H₃₇N₄O₄P·2/5CH₂O₂

Appearance

Solid

Color

White to off-white

SMILES

O=CO.O=P([C@@H](N)CCC1=CC=CC=C1)(O)C[C@H](CC(C)C)C(N[C@H](C(N)=O)CC2=CNC3=CC=CC=C23)=O.[0.4]

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : 50 mg/mL (94.16 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	1.8833 mL	9.4164 mL	18.8327 mL
5 mM	0.3767 mL	1.8833 mL	3.7665 mL
10 mM	0.1883 mL	0.9416 mL	1.8833 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Molarity Calculator
Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)

Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Data Sheet (272 KB) SDS (251 KB) Handling Instructions (2659 KB)

References

[1]. Birgit Wilding, et al. Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1. Bioorg Med Chem Lett. 2021 Jun 15;42:128050. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	1.8833 mL	9.4164 mL	18.8327 mL	47.0819 mL
	5 mM	0.3767 mL	1.8833 mL	3.7665 mL	9.4164 mL
	10 mM	0.1883 mL	0.9416 mL	1.8833 mL	4.7082 mL
	15 mM	0.1256 mL	0.6278 mL	1.2555 mL	3.1388 mL
	20 mM	0.0942 mL	0.4708 mL	0.9416 mL	2.3541 mL
	25 mM	0.0753 mL	0.3767 mL	0.7533 mL	1.8833 mL
	30 mM	0.0628 mL	0.3139 mL	0.6278 mL	1.5694 mL
	40 mM	0.0471 mL	0.2354 mL	0.4708 mL	1.1770 mL
	50 mM	0.0377 mL	0.1883 mL	0.3767 mL	0.9416 mL
	60 mM	0.0314 mL	0.1569 mL	0.3139 mL	0.7847 mL
	80 mM	0.0235 mL	0.1177 mL	0.2354 mL	0.5885 mL

DG013B formate Related Classifications

Others

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DG013B formateAminopeptidaseInhibitorinhibitorinhibit

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