1. GPCR/G Protein
    Neuronal Signaling
    Immunology/Inflammation
  2. Histamine Receptor
  3. Samelisant free base

Samelisant free base (Synonyms: SUVN-G3031 free base)

Cat. No.: HY-122608
Handling Instructions

Samelisant (SUVN-G3031) free base is a selective inverse agonist at Histamine 3 receptor (H3R) whose Ki value towards hH3R is 8.73 nM. Samelisant has adequate oral exposures and favorable elimination half-lives both in rats and dogs.

For research use only. We do not sell to patients.

Samelisant free base Chemical Structure

Samelisant free base Chemical Structure

CAS No. : 1394808-82-2

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Description

Samelisant (SUVN-G3031) free base is a selective inverse agonist at Histamine 3 receptor (H3R) whose Ki value towards hH3R is 8.73 nM. Samelisant has adequate oral exposures and favorable elimination half-lives both in rats and dogs[1][2].

Molecular Weight

373.49

Formula

C₂₁H₃₁N₃O₃

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Samelisant free base
Cat. No.:
HY-122608
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