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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
9 Results for "
CDK9/CycT
" in MedChemExpress (MCE) Product Catalog:
Products (9)
9 Results for "CDK9/CycT" in MCE Product Catalog:
41
41 Publications Verification
NVP-2 is a potent and selective ATP-competitive cyclin dependent kinase 9 (CDK9) probe, inhibits CDK9/CycT activity with an IC50 of 0.514 nM. NVP-2 displays inhibitory effcts on CDK1/CycB, CDK2/CycA and CDK16/CycY kinases with IC50 values of 0.584 μM, 0.706 μM, and 0.605 μM, respectively. NVP-2 induces cell apoptosis.
10
10 Cited Publications
Synonyms: BAY-1143572
Atuveciclib (BAY-1143572) is a potent and highly selective, oral PTEFb/CDK9 inhibitor. Atuveciclib (BAY-1143572) inhibits CDK9/CycT1 with an IC50 of 13 nM .
1
1 Cited Publications
Synonyms: BAY-1143572 Racemate
Atuveciclib Racemate (BAY-1143572 Racemate) is the racemate mixture of Atuveciclib. Atuveciclib is a potent and highly selective, oral P-TEFb/CDK9 inhibitor which supresses CDK9/CycT1 with an IC50 of 13 nM.
1
Synonyms: BAY-1143572 S-Enantiomer; (+)-Atuveciclib; (+)-BAY-1143572
Atuveciclib S-Enantiomer (BAY-1143572 S-Enantiomer) is a potent and selective CDK9 inhibitor, which inhibits CDK9/CycT1 with an IC50 of 16 nM.
Cat. No.: HY-156795
CAS No.: 3020773-91-2
PROTAC CDK9/CycT1 Degrader-2 is a inhibitor of CDK9, with the IC50 of 45 nM .
Cat. No.: HY-156083
CAS No.: 3020773-81-0
PROTAC CDK9/CycT1 Degrader-1 (compounds 10) is a potent inhibitor of CDK9. PROTAC CDK9/CycT1 Degrader-1 can be used as a PROTAC target protein ligand for PROTAC synthesis. PROTAC CDK9/CycT1 Degrader-1 shows strong anti-proliferative activity in solid tumors .
Cat. No.: HY-13231R
CAS No.: 1415559-43-1
CDK9-IN-1 (Standard) is the analytical standard of CDK9-IN-1. This product is intended for research and analytical applications. CDK9-IN-1 is a novel, selective CDK9 inhibitor for the treatment of HIV infection, with an IC50 of 39 nM for CDK9/CycT1, extracted from reference, compound 87.
Cat. No.: HY-P703098
Purity: ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: CCNT1; Cyclin-T1; Prev. HIVE1; Cyclin C-Related Protein; CycT1; MLLT10/CCNT1 Fusion; CCNT; Cyclin-T; Human Immunodeficiency Virus Type 1 (HIV-1) Expression (Elevated) 1; CycT1; Cyclin T1; CDK9-Associated C-Type Protein
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
