PROTAC CDK9/CycT1 Degrader-2
PROTAC CDK9/CycT1 Degrader-2 is a inhibitor of CDK9, with the IC50 of 45 nM.
For research use only. We do not sell to patients.
- CAS No.: 3020773-91-2
- Formula: C30H36N4O6S2
- Molecular Weight:612.76
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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CDK9 45 nM (IC50) |
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| U2932 | IC50 |
45 nM
Compound: 16
|
Cytotoxicity against human U2932 cells assessed as inhibition of cell growth measured after 72 hrs by CCK-8 assay
Cytotoxicity against human U2932 cells assessed as inhibition of cell growth measured after 72 hrs by CCK-8 assay
|
[PMID: 37671907] |
Chemical Information
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CAS No. 3020773-91-2
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Molecular Weight 612.76
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Formula C30H36N4O6S2
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SMILES
O=C1OC2=CC(OCCCN3CCC(CC3)C(NC4=NC=C(S4)SCC5=NC=C(O5)C(C)(C)C)=O)=CC(O)=C2C(C)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)