8 Results for "

Gemfibrozil

" in MedChemExpress (MCE) Product Catalog:
Products (8)

8 Results for "Gemfibrozil" in MCE Product Catalog:

6
6 Cited Publications
Cat. No.: HY-B0258
CAS No.: 25812-30-0
Synonyms: CI-719
Gemfibrozil is an activator of PPAR-α, used as a lipid-lowering agent; Gemfibrozil is also a nonselective inhibitor of several P450 isoforms, with Ki values for CYP2C9, 2C19, 2C8, and 1A2 of 5.8, 24, 69, and 82 μM, respectively.
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1
1 Cited Publications
Cat. No.: HY-129993
CAS No.: 91683-38-4
Purity:  98.79%
Gemfibrozil 1-O-β-Glucuronide, a metabolite of Gemfibrozil (CI-719; HY-B0258), is a potent and competitive P450 (CYP) isoform CYP2C8 inhibitor with an IC50 of 4.07 μM .
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Cat. No.: HY-B0258R
CAS No.: 25812-30-0
Synonyms: CI-719 (Standard)
Gemfibrozil (Standard) is the analytical standard of Gemfibrozil. This product is intended for research and analytical applications. Gemfibrozil is an activator of PPAR-α, used as a lipid-lowering agent; Gemfibrozil is also a nonselective inhibitor of several P450 isoforms, with Ki values for CYP2C9, 2C19, 2C8, and 1A2 of 5.8, 24, 69, and 82 μM, respectively.
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Cat. No.: HY-B0258S
CAS No.: 1184986-45-5
Synonyms: CI-719-d6
Gemfibrozil-d6 is the deuterium labeled Gemfibrozil. Gemfibrozil is an activator of PPAR-α, used as a lipid-lowering agent; Gemfibrozil is also a nonselective inhibitor of several P450 isoforms, with Ki values for CYP2C9, 2C19, 2C8, and 1A2 of 5.8, 24, 69, and 82 μM, respectively.
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Cat. No.: HY-W699866
CAS No.: 1703747-47-0
Gemfibrozil 1-O-β-glucuronide-d6 is the deuterium labeled Gemfibrozil 1-O-β-glucuronide (HY-129993). Gemfibrozil 1-O-β-Glucuronide, a metabolite of Gemfibrozil (CI-719; HY-B0258), is a potent and competitive P450 (CYP) isoform CYP2C8 inhibitor with an IC50 of 4.07 μM .
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Cat. No.: HY-B0258S1
CAS No.: 1160569-36-7
Synonyms: CI-719-d6-1
Gemfibrozil-d6-1 (CI-719-d6-1) is the deuterium labeled Gemfibrozil (HY-B0258). Gemfibrozil is an activator of PPAR-α, used as a lipid-lowering agent; Gemfibrozil is also a nonselective inhibitor of several P450 isoforms, with Ki values for CYP2C9, 2C19, 2C8, and 1A2 of 5.8, 24, 69, and 82 μM, respectively .
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Cat. No.: HY-173014
CAS No.: 2396744-05-9
Research Areas:  

Metabolic Disease

Gemfibrozil glucoside (Compound 4n) is a glycoside based on Gemfibrozil (HY-B0258). Gemfibrozil glucoside has lipid-lowering effects .
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Cat. No.: HY-E72113
Target:  

UGT

Research Areas:  

Cardiovascular Disease

Human UGT2B7 is a UDP-glucuronosyltransferase isoform. Human UGT2B7 catalyzes the glucuronidation of Clopidogrel carboxylic acid (HY-141749A), Chloramphenicol (HY-B0239), and Morphine. Human UGT2B7 can be used in studies related to acute coronary syndrome and thrombus-induced events .
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