5 Results for "

KOPR

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "KOPR" in MCE Product Catalog:

Cat. No.: HY-110252
CAS No.: 92545-30-7
Purity:  ≥99.0%
Salvinorin B is a selective and brain-penetrant kappa opioid receptor (KOPr) agonist with an EC50 of 248 nM and Ki of 2.95 μM. Salvinorin B activates downstream signaling pathways by binding to KOPr, inhibits pain transmission and reduces inflammatory response. Salvinorin B can be used for the researches of inflammation, immunology and neurological disease, such as neuropathic pain, multiple sclerosis and anxiety .
loading...
    loading...
Cat. No.: HY-100845
CAS No.: 83729-01-5
Synonyms: Divinorin A
Salvinorin A is a potent, unique and short-acting high efficacy kappa-opioid receptor (KOPr) agonist with Ki value of 4.3 nm. Salvinorin A is a non-nitrogenous neoclerodane isolated from Salvia divinorum.
loading...
    loading...
Cat. No.: HY-135230
CAS No.: 1346133-11-6
Purity:  99.59%
Synonyms: FP3FBZ
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

LY2444296 is an orally bioavailable, high-affinity and selective short-acting kappa opioid receptor (KOPR) antagonist, with a Ki value of ~1 nM. LY2444296 exhibits anti-anxiety like effects .
loading...
    loading...
Cat. No.: HY-137920
CAS No.: 689295-71-4
Target:  

Opioid Receptor

Research Areas:  

Cardiovascular Disease

Salvinorin A (Divinorin A) propionate is a potent, unique and short-acting high efficacy kappa-opioid receptor (KOPr) agonist with Ki value of 4.3 nm. Salvinorin A propionate is a non-nitrogenous neoclerodane isolated from Salvia divinorum .
loading...
    loading...
Cat. No.: HY-126910
CAS No.: 862073-79-8
Target:  

Opioid Receptor

Research Areas:  

Metabolic Disease

Mesyl Salvinorin B is a potent and selective kappa opioid receptor (KOP-r) agonist. Mesyl Salvinorin B prevents the ADE (Alcohol deprivation effect) in mice. Mesyl Salvinorin B dose-dependently reduces alcohol intake and preference in CED (chronic escalation drinking) mice .
loading...
    loading...