11 Results for "

cyclic amide

" in MedChemExpress (MCE) Product Catalog:
Products (11)

11 Results for "cyclic amide" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-19469
CAS No.: 359625-79-9
Synonyms: CYR-101; MIN-101; MT-210
Research Areas:  

Neurological Disease

Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively).
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1
1 Cited Publications
Cat. No.: HY-P3929A
CAS No.: 1293946-39-0
Target:  

PKA

Research Areas:  

Cancer

PKI (14-24)amide TFA is a potent PKA inhibitor. PKI (14-24)amide strongly inhibited cyclic AMP-dependent protein kinase activity in the cell homogenate .
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Cat. No.: HY-Y1275
CAS No.: 872-50-4
Synonyms: NMP; 1-Methyl-2-pyrrolidinone
N-Methylpyrrolidone (1-Methyl-2-pyrrolidinone), a five-membered cyclic amide, is an orally active organic polar solvent with teratogenicity and toxicity. N-Methylpyrrolidone is low in acute toxicity with a LD50 value of 3914 mg/kg in rats and of 4050 mg/kg in mice. N-Methylpyrrolidone is extensively used in the manufacture of adhesives, paints, fuels, and pharmaceuticals .
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Cat. No.: HY-Y1275S
CAS No.: 185964-60-7
Synonyms: NMP-d9; 1-Methyl-2-pyrrolidinone-d9
N-Methylpyrrolidone-d9 (NMP-d9) is deuterium labeled N-Methylpyrrolidone. N-Methylpyrrolidone (1-Methyl-2-pyrrolidinone), a five-membered cyclic amide, is an orally active organic polar solvent with teratogenicity and toxicity. N-Methylpyrrolidone is low in acute toxicity with a LD50 value of 3914 mg/kg in rats and of 4050 mg/kg in mice. N-Methylpyrrolidone is extensively used in the manufacture of adhesives, paints, fuels, and pharmaceuticals .
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Cat. No.: HY-W251708
CAS No.: 91713-91-6
Target:  

Endogenous Metabolite

Research Areas:  

Neurological Disease

AHR 10240, a cyclic amide, is a metabolite of Bromfenac (HY-B1888). AHR 10240 can be used for analgesia research
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Cat. No.: HY-Y1275S1
CAS No.: 933-86-8
Synonyms: NMP-d3; N-Methyl-2-pyrrolidone-d3
N-Methylpyrrolidone-d3 is the deuterium labeled N-Methylpyrrolidone . N-Methylpyrrolidone (1-Methyl-2-pyrrolidinone), a five-membered cyclic amide, is an organic polar solvent. N-Methylpyrrolidone is extensively used in the manufacture of adhesives, paints, fuels, and pharmaceuticals .
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Cat. No.: HY-E70077
CAS No.: 9001-74-5
Target:  

Endogenous Metabolite

Research Areas:  

Infection Metabolic Disease

Penicillinase (from calf stomach) is an enzyme that degrades penicillin by hydrolyzing the cyclic amide bonds in the lactam ring of penicillin, which can inactivate penicillin. Penicillinase (from calf stomach) can be isolated from penicillin resistant strains. Penicillinase (from calf stomach) has potential application as a marker for steroid hormone enzyme linked immunosorbent assay .
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Cat. No.: HY-P3929
CAS No.: 100853-61-0
Target:  

PKA

Research Areas:  

Cancer

PKI (14-24)amide is a potent PKA inhibitor. PKI (14-24)amide strongly inhibited cyclic AMP-dependent protein kinase activity in the cell homogenate .
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Cat. No.: HY-P3785
CAS No.: 100853-58-5
Target:  

PKA

Research Areas:  

Neurological Disease

PKI(5-22)amide is the active inhibitory fragment of the inhibitor of the cyclic AMP-dependent protein kinase (PKA). PKI(5-22)amide inhibits PKA activation, but fails to attenuate homologous desensitization of CRF1 receptors .
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Cat. No.: HY-W976179
CAS No.: 42997-42-2
2E,4E-Decadienoylpiperidide (Compound 2) is a cyclic amide compound that can be found in the roots, leaves, and flowers of Achillea ptarmica .
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Cat. No.: HY-E71344
Research Areas:  

Others

γ-L-Glutamyl-butirosin B γ-Glutamyl cyclotransferase (EC 4.3.2.6) catalyses the last step in the biosynthesis of the aminoglycoside antibiotic butirosin B. The enzyme acts as a cyclotransferase, cleaving the amide bond via transamidation using the α-amine of the terminal γ-L-glutamate of the side chain, releasing it as the cyclic 5-oxoproline.
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