1. GPCR/G Protein
    Neuronal Signaling
  2. Adrenergic Receptor
  3. Terazosin

Terazosin 

Cat. No.: HY-B0371
Handling Instructions

Terazosin is a quinazoline derivative and a competitive and orally active α1-adrenoceptor antagonist. Terazosin works by relaxing blood vessels and the opening of the bladder. Terazosin has the potential for benign prostatic hyperplasia (BPH) and high blood pressure treatment.

For research use only. We do not sell to patients.

Terazosin Chemical Structure

Terazosin Chemical Structure

CAS No. : 63590-64-7

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Description

Terazosin is a quinazoline derivative and a competitive and orally active α1-adrenoceptor antagonist. Terazosin works by relaxing blood vessels and the opening of the bladder. Terazosin has the potential for benign prostatic hyperplasia (BPH) and high blood pressure treatment[1][2][3].

IC50 & Target

α1-adrenoceptor[1]

In Vitro

Terazosin does not discriminate cloned α1-adrenoceptor subtypes transiently expressed in COS cells[1].

In Vivo

Terazosin can be used to promote stone discharge in treatment of ureteral stones. Terazosin is reportedly safe and effective in treatment of distal ureteral stones, especially stones >5 mm[3].

Clinical Trial
Molecular Weight

387.43

Formula

C₁₉H₂₅N₅O₄

CAS No.

63590-64-7

SMILES

O=C(N1CCN(C2=NC(N)=C3C=C(OC)C(OC)=CC3=N2)CC1)C4OCCC4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

TerazosinAdrenergic ReceptorBeta Receptorα1-adrenoceptorbenignprostatichyperplasiahighbloodpressurebladderquinazolineInhibitorinhibitorinhibit

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Terazosin
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